Table 6: Summary of modulators

ReceptorChannel modulator
iGluR1 flipCyclothiazide (CTZ)
iGluR1 flopLY compound
iGluR4 flipCyclothiazide (CTZ)
iGluR4 flopLY compound
iGluR5 & 6Concanavalin A (Con A)

From: FLIPRâ„¢ Assays for GPCR and Ion Channel Targets

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Assay Guidance Manual [Internet].
Sittampalam GS, Gal-Edd N, Arkin M, et al., editors.
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