CID/ML#Target NameIC50/EC50 (nM) [SID, AID]Anti-target Name(s)IC50/EC50 (μM) [SID, AID]SelectivitySecondary Assay(s) Name: IC50/EC50 (nM) [SID, AID]
CID 44191096 ML128mGluR4240 (hm) 110 (rat) [SID-85240643, AID-2185, AID-2197]mGluRs 1,2,3,5,7, 8 PanLabs> 10 μM [SID-85240643, AID-2193, AID-2191, AID-2190, AID-2188, AID-2183, AID-2182, AID-2181]>50Fold-Shift 28x(hm), 35x(rat)

[SID-85240643, AID-2179, AID-2180]

From: Discovery of a potent, selective and in vivo active mGluR4 positive allosteric modulator

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Probe Reports from the NIH Molecular Libraries Program [Internet].

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