Table 4SAR and Selectivity

Compound IDAssay FormatAssay TargetNo of RunsIC50 Value (μM)
MLS-0014097LuminescentTNAP4>100
MLS-0014097LuminescentPLAP~ 62.34
MLS-0014097LuminescentIAP120.7
MLS-0014097ColorimetricGAPDH2>100
MLS-0014097FPBCL-b/TR31>100
MLS-0014097FPBfl-11>100

From: Placental Alkaline Phosphatase (PLAP) Luminescent HTS assay - Probe 1

Cover of Probe Reports from the NIH Molecular Libraries Program
Probe Reports from the NIH Molecular Libraries Program [Internet].

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