AIDTargetConcentrationBioassay type
1631hPKM2 Activator57 μM to 0.4 nMPrimary qHTS
1634hPKM2 Inhibitor57 μM to 0.4 nMPrimary qHTS
1540hPKM257 μM to 0.4 nMConfirmatory
1541hPKL57 μM to 0.4 nMSelectivity
1542hPKM157 μM to 0.4 nMSelectivity
1543hPKR57 μM to 0.4 nMSelectivity

From: Identification of activators for the M2 isoform of human pyruvate kinase

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