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3BWJ:
Complex of PKA with the bisubstrate protein kinase inhibitor lead compound Arc-1034
PDB ID:
3BWJ
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MMDB ID:
69396
PDB Deposition Date:
2008/1/9
Updated in MMDB:
2017/11
Experimental Method:
x-ray diffraction
Resolution:
2.3 Å
Source Organism:
Bos taurus
Similar Structures:
VAST+
Download sequence data
Biological Unit for 3BWJ: monomeric; determined by author and by software (PISA)
Molecular Components in 3BWJ
Label
Count
Molecule
Protein (1 molecule)
A
1
Camp-dependent Protein Kinase, Alpha-catalytic Subunit
(Gene symbol:
PRKACA
)
Chemicals and Non-standard biopolymers (2 molecules)
1
2
(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-(6-{[(1R)-4-carbamimidamido-1-{[(1R)-4-carbamimidamido-1-carbamoylbutyl]carbamoyl}butyl]amino}-6-oxohexyl)-3,4-dihydroxytetrahydrofuran-2-carboxamide
* Click molecule labels to explore molecular sequence information.
Citing MMDB
Madej T, Lanczycki CJ, Zhang D, Thiessen PA, Geer RC, Marchler-Bauer A, Bryant SH.
"
MMDB and VAST+: tracking structural similarities between macromolecular complexes.
Nucleic Acids Res. 2014 Jan; 42(Database issue)
:D297-303